SCHEMBL4726796

SCHEMBL4726796

CC(C)(C)c1cc(CBr)cc(C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 8/20 0.46
RXRB P28702 8/20 0.46
RXRG P48443 4/20 0.46
FOLH1 Q04609 1/20 0.43
NR1H4 Q96RI1 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
MAPK1 P28482 1/20 0.42
BLM P54132 1/20 0.42
CASP7 P55210 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SRD5A2 P31213 1/20 0.42
EPHX2 P34913 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.40
NR4A2 P43354 2/20 0.40
NR4A1 P22736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10235447 0.84 RXRA (0.47) RXRARXRBRXRGFOLH1NR1H4
SCHEMBL545316 0.84 RXRA (0.47) RXRARXRBRXRGFOLH1NR1H4
SCHEMBL5335840 0.81 NOTUM (0.46) TDP1
SCHEMBL166878 0.80 RXRB (0.59) RXRARXRBRXRGNR1H4TDP1
SCHEMBL501957 0.80 RXRB (0.64) RXRARXRBRXRGNR1H4TDP1
SCHEMBL2226759 0.80 TTR (0.44) RXRARXRBFOLH1TDP1TP53
SCHEMBL1866724 0.80 TTR (0.44) FOLH1TDP1TP53MAPTALOX15
Acetic Acid SCHEMBL28155950 0.79 TPMT (0.43) RXRARXRBFOLH1TDP1TP53
Hydrochloric Acid SCHEMBL4585979 0.78 RXRB (0.57) RXRARXRBRXRGNR1H4TDP1
Hydrochloric Acid SCHEMBL11879619 0.78 RXRB (0.57) RXRARXRBRXRGNR1H4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed