SCHEMBL4727756

SCHEMBL4727756

[CH2]CCC(C)Nc1cc(OC)cc2ccc(C(C)(C)C)nc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
KDM4E B2RXH2 3/20 0.48
CYP1A2 P05177 2/20 0.48
CASP1 P29466 2/20 0.48
ALDH1A1 P00352 2/20 0.48
LMNA P02545 2/20 0.48
TP53 P04637 2/20 0.48
ABCB11 O95342 1/20 0.48
ESR1 P03372 1/20 0.48
PGR P06401 1/20 0.48
ADRB2 P07550 1/20 0.48
CHRM2 P08172 1/20 0.48
ADRB1 P08588 1/20 0.48
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
NQO2 P16083 1/20 0.48
MAOA P21397 1/20 0.48
PTGS1 P23219 1/20 0.48
SLC6A2 P23975 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5080647 0.86 MAOA (0.66) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL4727369 0.80 KDM4E (0.48) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL6268435 0.79 KDM4E (0.47) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL6280385 0.79 HSP90AA1 (0.48) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL6280393 0.79 HSP90AA1 (0.48) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL4727368 0.79 HSP90AA1 (0.48) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL5083237 0.78 IDO1 (0.47) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL6276764 0.77 KDM4E (0.46) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL5086463 0.77 HSP90AA1 (0.51) IDO1KDM4ECYP1A2CASP1ALDH1A1
SCHEMBL5086470 0.77 HSP90AA1 (0.46) IDO1KDM4ECYP1A2CASP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021210-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-02-21 WO disclosed