SCHEMBL4728056

SCHEMBL4728056

COc1cc2ncn(C3CC3)c(=O)c2cc1OCCc1ccc2ccccc2n1

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.47
CYP1A2 P05177 1/20 0.47
HCRTR1 O43613 6/20 0.45
HCRTR2 O43614 6/20 0.45
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
HDAC6 Q9UBN7 2/20 0.41
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4794353 0.96 PDE10A (0.46) PDE10ACYP1A2HCRTR1HCRTR2BCHE
SCHEMBL4727776 0.96 PDE10A (0.46) PDE10ACYP1A2HCRTR1HCRTR2BCHE
SCHEMBL4729965 0.86 HDAC6 (0.47) PDE10ACYP1A2HCRTR1HCRTR2HDAC6
SCHEMBL4729821 0.85 PDE10A (0.48) PDE10ACYP1A2HCRTR1HCRTR2HDAC6
SCHEMBL4729506 0.84 HDAC6 (0.49) PDE10ACYP1A2HDAC6ADRA1AADRA1B
SCHEMBL4726934 0.83 HDAC6 (0.45) PDE10ACYP1A2HDAC6
SCHEMBL4728780 0.83 PDE10A (0.46) PDE10ACYP1A2HCRTR1HCRTR2BCHE
SCHEMBL4725564 0.83 HDAC6 (0.44) PDE10ACYP1A2HCRTR1HCRTR2HDAC6
SCHEMBL4781644 0.78 IRAK1 (0.52) HDAC6
SCHEMBL4725230 0.74 ACHE (0.55) PDE10AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO claimed