SCHEMBL4781644

SCHEMBL4781644

COc1cc2ncn(C3CC3)c(=O)c2cc1OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IRAK1 P51617 1/20 0.52
IRAK4 Q9NWZ3 1/20 0.52
HDAC6 Q9UBN7 2/20 0.49
ELANE P08246 1/20 0.48
PDE4B Q07343 1/20 0.48
KIT P10721 2/20 0.46
PLK1 P53350 2/20 0.46
KDR P35968 1/20 0.46
CTSV O60911 2/20 0.46
CTSL P07711 2/20 0.46
EGFR P00533 1/20 0.46
KDM1A O60341 1/20 0.45
CHRNA7 P36544 2/20 0.45
TLR9 Q9NR96 2/20 0.45
TLR7 Q9NYK1 2/20 0.45
NSD2 O96028 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19645656 0.83 ELANE (0.53) IRAK1IRAK4HDAC6ELANEKIT
SCHEMBL17192046 0.81 KIT (0.41) HDAC6KITPLK1KDRCTSL
SCHEMBL6879935 0.80 HDAC6 (0.78) HDAC6ELANEPLK1EGFR
SCHEMBL4725517 0.80 ELANE (0.50) IRAK1IRAK4HDAC6ELANEPDE4B
SCHEMBL4728056 0.78 PDE10A (0.47) HDAC6
SCHEMBL4594235 0.77 HDAC6 (0.68) HDAC6
SCHEMBL4796792 0.77 HDAC6 (0.48) HDAC6EGFR
SCHEMBL7121138 0.76 KIT (0.48) IRAK1IRAK4ELANEKITKDR
SCHEMBL663991 0.76 HDAC6 (0.54) HDAC6ELANEPLK1EGFRTLR9
SCHEMBL4300106 0.76 HDAC6 (0.60) HDAC6EGFRTLR9TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed