SCHEMBL4728679

SCHEMBL4728679

COc1ccc(-c2ncnc3cc(OCc4ccccc4)ccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 3/20 0.56
NPSR1 Q6W5P4 3/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
EGFR P00533 3/20 0.53
ERBB2 P04626 1/20 0.51
TLR8 Q9NR97 1/20 0.50
MAOB P27338 1/20 0.50
MAPT P10636 3/20 0.48
MAPK1 P28482 1/20 0.47
NOD2 Q9HC29 1/20 0.47
MEN1 O00255 1/20 0.47
KDR P35968 1/20 0.47
KMT2A Q03164 1/20 0.47
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CAMKK1 Q8N5S9 1/20 0.46
CAMKK2 Q96RR4 1/20 0.46
PRMT5 O14744 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728722 0.91 ADORA2A (0.53) KITEGFRERBB2TLR8MAOB
SCHEMBL4727883 0.86 CYP3A4 (0.49) KITEGFRERBB2TLR8MAOB
SCHEMBL4730192 0.82 PDE10A (0.55)
SCHEMBL4727924 0.81 MAPT (0.49) KITALDH1A1LMNATLR8MAPT
SCHEMBL28872954 0.78 ADORA2A (0.66) NPSR1ALDH1A1LMNAHTTEGFR
SCHEMBL4725258 0.77 KDM1A (0.57) KITLMNAHTTEGFRMAPK1
SCHEMBL6824579 0.77 PRMT5 (0.50) NPSR1ALDH1A1LMNAHTTEGFR
SCHEMBL7982589 0.77 CSF1R (0.57) KITEGFRERBB2MAOBMAPT
SCHEMBL4725570 0.76 IP6K1 (0.50) EGFRERBB2PRMT5CYP3A4FLT3
SCHEMBL5465811 0.76 MEN1 (0.55) KITLMNAEGFRERBB2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed