SCHEMBL4729066

SCHEMBL4729066

COc1cccc(CNC(=O)c2ccc(-c3cc(NC(=O)c4cc(C(C)(C)C)ccc4OC)cnc3C)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.50
ROCK1 Q13464 7/20 0.50
PRKACA P17612 2/20 0.50
PRKX P51817 2/20 0.50
PRKCQ Q04759 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
MMP13 P45452 2/20 0.49
MAPK14 Q16539 2/20 0.47
MAPK11 Q15759 1/20 0.47
PDGFRB P09619 1/20 0.46
FLT4 P35916 1/20 0.46
GRK5 P34947 1/20 0.46
TP53 P04637 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4729418 0.93 MEN1 (0.44) ROCK2ROCK1PRKACAPRKXPRKCQ
SCHEMBL4729229 0.90 MEN1 (0.52) ROCK2
SCHEMBL4727856 0.88 MEN1 (0.45) CYP3A4L3MBTL1
SCHEMBL4781615 0.85 HPGD (0.51) ROCK2ROCK1TP53
SCHEMBL4727301 0.82 STIM1 (0.46) TP53
SCHEMBL4727417 0.80 STIM1 (0.44)
SCHEMBL4727073 0.79 MAPK14 (0.48) MAPK14MAPK11
SCHEMBL4728221 0.78 HPGD (0.48) ROCK2CYP2C9MAPK14L3MBTL1
SCHEMBL4727373 0.76 RAF1 (0.47) MAPK14
SCHEMBL4782260 0.76 MEN1 (0.51) ROCK2ROCK1CYP3A4MMP13MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed