SCHEMBL4729443

SCHEMBL4729443

CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC[C@H]4CCCC(N)(N)[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.65
CYP2C19 P33261 1/20 0.65
INPP5D Q92835 1/20 0.64
CDC25A P30304 5/20 0.54
POLA1 P09884 1/20 0.53
CDC25B P30305 1/20 0.53
SRD5A1 P18405 4/20 0.53
SRD5A2 P31213 3/20 0.53
FNTA P49354 2/20 0.50
FNTB P49356 2/20 0.50
NPC1L1 Q9UHC9 2/20 0.50
AKR1B10 O60218 1/20 0.50
AKR1B1 P15121 1/20 0.50
EFNA1 P20827 1/20 0.50
EPHA2 P29317 1/20 0.50
PSEN1 P49768 1/20 0.50
PSEN2 P49810 1/20 0.50
GPBAR1 Q8TDU6 1/20 0.50
APH1B Q8WW43 1/20 0.50
NCSTN Q92542 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4728585 0.99 INPP5D (0.66) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL28057976 0.89 CYP2D6 (0.62) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL7514775 0.87 CYP2D6 (0.62) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL9664069 0.87 CYP2D6 (0.62) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL15346210 0.87 CYP2D6 (0.62) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL28959940 0.83 CYP2D6 (0.58) CYP2D6CYP2C19INPP5DCDC25APOLA1
Methylamine SCHEMBL27360770 0.83 CYP2D6 (0.72) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL135273 0.83 CYP2D6 (0.71) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL19866272 0.83 CYP2D6 (0.71) CYP2D6CYP2C19INPP5DCDC25APOLA1
SCHEMBL14676689 0.83 CYP2D6 (0.71) CYP2D6CYP2C19INPP5DCDC25APOLA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008038965-A1 7ALPHA-AMINOSTEROID DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PREPARATION METHOD THEREOF AND COMPOSITION FOR ANTICANCER OR ANTIBIOTICS CONTAINING THE SAME AS AN ACTIVE INGREDIENT KYUNGPOOK NATIONAL UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2008-04-03 WO claimed
WO-2008038965-A1 7ALPHA-AMINOSTEROID DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PREPARATION METHOD THEREOF AND COMPOSITION FOR ANTICANCER OR ANTIBIOTICS CONTAINING THE SAME AS AN ACTIVE INGREDIENT KYUNGPOOK NATIONAL UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2008-04-03 WO disclosed