SCHEMBL4732010

SCHEMBL4732010

CC1(C(=O)NCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CCN(C(=O)O)CC1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 11/20 0.51
TACR1 P25103 2/20 0.50
CCR5 P51681 1/20 0.47
CYP3A4 P08684 3/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
USP2 O75604 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.45
MTOR P42345 1/20 0.45
KCNH2 Q12809 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13222832 0.89 CYP2D6 (0.48) CCR2TACR1CCR5CYP3A4ALDH1A1
SCHEMBL3036649 0.86 CCR2 (0.49) CCR2TACR1CCR5CYP3A4ALDH1A1
SCHEMBL3040315 0.85 TACR1 (0.55) CCR2TACR1CCR5CYP3A4ALDH1A1
SCHEMBL13243692 0.83 CCR2 (0.43) CCR2TACR1CCR5CYP3A4ALDH1A1
SCHEMBL3030595 0.81 CCR2 (0.48) CCR2TACR1CCR5CYP3A4ALDH1A1
SCHEMBL14221691 0.81 TACR1 (0.65) CCR2TACR1CYP3A4ALDH1A1TSHR
SCHEMBL3997558 0.81 CCR2 (0.51) CCR2TACR1KCNH2
Ammonia Solution, Strong SCHEMBL3036646 0.80 TACR1 (0.64) CCR2TACR1CYP3A4ALDH1A1TSHR
Trifluoroacetic Acid SCHEMBL3030594 0.80 TACR1 (0.64) CCR2TACR1CYP3A4ALDH1A1CYP2D6
SCHEMBL3042038 0.77 CCR2 (0.55) CCR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008045564-A2 CARBOXAMIDE COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE CHEMOKINE CCR2 RECEPTOR EPIX DELAWARE, INC. (US) 2008-04-17 WO disclosed