SCHEMBL4733058

SCHEMBL4733058

CS(=O)(=O)Nc1cc(CN(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)C(=O)C2(CC3CC3)CCNC2)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.36
TACR1 P25103 6/20 0.34
NR3C1 P04150 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731394 0.94 TRPV1 (0.42) TRPV1
SCHEMBL4730403 0.89 TACR1 (0.35) TACR1
SCHEMBL4733037 0.86 KCNH2 (0.41) TACR1
SCHEMBL4730021 0.86 TACR1 (0.38) TACR1
SCHEMBL4732027 0.84 TACR1 (0.38) TACR1
SCHEMBL4729164 0.84 TACR1 (0.35) TACR1
SCHEMBL4730989 0.84 CETP (0.38) TACR1
SCHEMBL4730613 0.83 TACR1 (0.35) TACR1
SCHEMBL4728683 0.82 KDM4E (0.40) TACR1
SCHEMBL4731956 0.81 TACR1 (0.46) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008045564-A2 CARBOXAMIDE COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE CHEMOKINE CCR2 RECEPTOR EPIX DELAWARE, INC. (US) 2008-04-17 WO disclosed