SCHEMBL4733239

SCHEMBL4733239

CN(c1ccc(NC(=O)Nc2cccc(C(F)(F)F)c2)cc1)c1ccnc(Cl)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.54
RIPK1 Q13546 3/20 0.54
MLKL Q8NB16 2/20 0.54
RIPK3 Q9Y572 2/20 0.54
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPT P10636 2/20 0.52
HTT P42858 1/20 0.52
RAB9A P51151 1/20 0.52
MAPK14 Q16539 5/20 0.52
TNNI3K Q59H18 5/20 0.52
BRAF P15056 3/20 0.52
TRPV1 Q8NER1 1/20 0.50
AURKA O14965 2/20 0.49
CSF1R P07333 1/20 0.49
PLK4 O00444 1/20 0.49
MAPK13 O15264 1/20 0.49
JAK2 O60674 1/20 0.49
MAP4K4 O95819 1/20 0.49
ABL1 P00519 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17979820 0.87 KDR (0.50) KDRRIPK1MLKLRIPK3BRAF
SCHEMBL17979914 0.84 KDR (0.49) KDRRIPK1MLKLRIPK3BRAF
SCHEMBL17260979 0.81 KDR (0.65) KDRRIPK1MLKLRIPK3MEN1
SCHEMBL23065786 0.80 KMT2A (0.62) KDRRIPK1MEN1KMT2AMAPT
SCHEMBL19899212 0.79 KDR (0.59) KDRRIPK1MLKLRIPK3MAPK14
SCHEMBL18024707 0.78 KDR (0.58) KDRRIPK1MLKLRIPK3MAPK14
SCHEMBL4733237 0.78 KMT2A (0.54) KDRRIPK1MEN1KMT2AMAPT
SCHEMBL4808894 0.77 POLB (0.47) KDRMEN1KMT2AMAPTHTT
SCHEMBL4735597 0.77 KDR (0.45) KDRMAPTRAB9AAURKANPC1
SCHEMBL4731171 0.76 KDR (0.61) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008060866-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-05-22 WO disclosed