SCHEMBL4733237

SCHEMBL4733237

O=C(Nc1ccc(NCc2ccnc(Cl)n2)cc1)Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54
KDR P35968 9/20 0.52
MAPK14 Q16539 7/20 0.52
TNNI3K Q59H18 7/20 0.52
BRAF P15056 6/20 0.52
TRPV1 Q8NER1 1/20 0.52
RIPK1 Q13546 1/20 0.51
CDK8 P49336 2/20 0.50
CDK7 P50613 1/20 0.50
CDK6 Q00534 1/20 0.50
PLK4 O00444 1/20 0.48
AURKA O14965 1/20 0.48
MAPK13 O15264 1/20 0.48
JAK2 O60674 1/20 0.48
MAP4K4 O95819 1/20 0.48
ABL1 P00519 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23065786 0.81 KMT2A (0.62) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL4733239 0.78 KDR (0.54) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL22155019 0.76 SMARCA2 (0.69) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL14601707 0.75 KMT2A (0.77) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL30101230 0.74 KMT2A (0.90) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL5597699 0.74 KMT2A (0.90) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL16654502 0.72 MAOA (0.56) KMT2AMAPTMEN1RAB9AJAK2
SCHEMBL17609423 0.72 MAPT (1.00) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL30069239 0.72 MAPT (1.00) KMT2AMAPTMEN1HTTRAB9A
SCHEMBL3260524 0.72 KDR (0.76) KMT2AMAPTMEN1HTTKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008060866-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-05-22 WO disclosed