SCHEMBL4734075

SCHEMBL4734075

Cc1nc(C(=O)O)cn1Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.57
NOTUM Q6P988 2/20 0.50
GAA P10253 1/20 0.45
PKM P14618 1/20 0.45
TSHR P16473 1/20 0.45
RIPK1 Q13546 1/20 0.45
POLB P06746 1/20 0.44
P2RX7 Q99572 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
P2RY14 Q15391 1/20 0.43
LMNA P02545 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4737901 0.92 BRD4 (0.51) BRD4NOTUMGAAPKMTSHR
SCHEMBL2360506 0.89 BRD4 (0.47) BRD4P2RY14ALDH1A1
SCHEMBL4024290 0.89 SMN1; SMN2 (0.47) BRD4NOTUMGAAPKMTSHR
SCHEMBL13363565 0.88 BRD4 (0.46) BRD4NOTUMGAARIPK1POLB
SCHEMBL16862950 0.88 BRD4 (0.59) BRD4NOTUMRIPK1P2RX7MEN1
SCHEMBL6799177 0.86 BRD4 (0.48) BRD4MEN1KMT2A
SCHEMBL17241086 0.85 P2RX7 (0.46) BRD4NOTUMPKMRIPK1P2RX7
SCHEMBL16862955 0.84 ALDH1A1 (0.60) GAATSHRP2RX7LMNAALDH1A1
SCHEMBL4419725 0.83 BRD4 (0.67) BRD4NOTUMGAAPKMTSHR
SCHEMBL4737896 0.80 BRD4 (0.41) BRD4NOTUMRIPK1P2RX7LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed