SCHEMBL4735982

SCHEMBL4735982

COc1c(C)cc(Br)cc1C.[MgH2]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
PKM P14618 1/20 0.44
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
HSD17B10 Q99714 2/20 0.41
ACHE P22303 1/20 0.39
ALDH1A1 P00352 4/20 0.38
NQO2 P16083 1/20 0.37
MAPT P10636 4/20 0.36
HTT P42858 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
TUBB4A P04350 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363341 0.97 KDM4E (0.45) KDM4EPKMCA2CA4HSD17B10
Hydrochloric Acid SCHEMBL28586799 0.95 KDM4E (0.44) KDM4EPKMCA2CA4HSD17B10
SCHEMBL11216824 0.85 HSD17B10 (0.52) KDM4EPKMCA2CA4HSD17B10
SCHEMBL11933625 0.83 ACHE (0.50) KDM4EPKMCA2CA4ACHE
SCHEMBL14394921 0.83 KDM4E (0.41) KDM4EPKMCA2CA4HSD17B10
SCHEMBL16904136 0.81 TDP1 (0.48) KDM4EPKMHSD17B10ALDH1A1MAPT
SCHEMBL931631 0.81 POLB (0.44) KDM4EPKMCA2CA4HSD17B10
SCHEMBL30017049 0.81 KDM4E (0.43) KDM4EPKMCA2CA4HSD17B10
SCHEMBL930657 0.81 KDM4E (0.40) KDM4EPKMCA2CA4HSD17B10
SCHEMBL19607300 0.81 KDM4E (0.43) KDM4EPKMCA2CA4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100548950-C Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2009-10-14 CN claimed
CN-1759084-A Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2006-04-12 CN claimed
CN-100548950-C Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2009-10-14 CN disclosed
CN-101391972-A Process of preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2009-03-25 CN disclosed
WO-2008070014-A2 BIARYL KETONE-SUBSTITUTED PIPERIDINES NEUROGEN CORPORATION (US) 2008-06-12 WO disclosed
CN-1759084-A Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2006-04-12 CN disclosed