SCHEMBL4735985

SCHEMBL4735985

CN(c1ccccc1)c1nc(C(=O)Cl)cs1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.53
NPC1 O15118 6/20 0.49
RAB9A P51151 5/20 0.49
KMT2A Q03164 3/20 0.49
HPGD P15428 2/20 0.49
TSHR P16473 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 2/20 0.49
NFKB1 P19838 2/20 0.49
NFKB2 Q00653 2/20 0.49
RELA Q04206 2/20 0.49
USP2 O75604 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
MAPK1 P28482 1/20 0.49
MMP13 P45452 1/20 0.49
HSD17B10 Q99714 1/20 0.49
GRIA1 P42261 1/20 0.43
CSNK2A2 P19784 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733657 0.88 CHEK1 (0.52) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL4739602 0.79 RAB9A (0.54) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL4734482 0.78 RAB9A (0.58) CHEK1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL11589312 0.75 NPC1 (0.48) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL11589491 0.75 HPGD (0.48) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL4762048 0.72 CHEK1 (0.41) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL9422086 0.71 NPC1 (0.80) NPC1RAB9AKMT2AHPGDTSHR
SCHEMBL13996099 0.70 NPC1 (0.49) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL3068359 0.70 LMNA (0.52) CHEK1NPC1RAB9AKMT2AHPGD
SCHEMBL168291 0.69 TDP1 (0.67) NPC1RAB9AKMT2AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed