SCHEMBL4736030

SCHEMBL4736030

CCN(CC)c1ccc(CN(C(=O)O)c2ccc(F)cc2)cn1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 2/20 0.47
AOC3 Q16853 1/20 0.44
LTB4R2 Q9NPC1 2/20 0.44
CNR2 P34972 5/20 0.42
CNR1 P21554 2/20 0.42
BCL2A1 Q16548 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPK14 Q16539 2/20 0.39
GBA1 P04062 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3071006 0.90 CACNA1H (0.47) CACNA1HAOC3LTB4R2CNR2BCL2A1
SCHEMBL3815393 0.87 CACNA1H (0.45) CACNA1HAOC3LTB4R2CNR2CNR1
SCHEMBL3064331 0.87 CACNA1H (0.45) CACNA1HAOC3LTB4R2CNR2BCL2A1
SCHEMBL3816063 0.86 CACNA1H (0.45) CACNA1HAOC3LTB4R2CNR2CNR1
SCHEMBL3825186 0.85 CACNA1H (0.44) CACNA1HAOC3LTB4R2CNR2CNR1
SCHEMBL3063271 0.85 RIPK1 (0.49) CACNA1HAOC3LTB4R2CNR2BCL2A1
Trifluoroacetic Acid SCHEMBL3054195 0.84 CACNA1H (0.42) CACNA1HAOC3LTB4R2CNR2CNR1
SCHEMBL3065942 0.84 CACNA1H (0.46) CACNA1HAOC3LTB4R2CNR2BCL2A1
SCHEMBL3821700 0.83 CNR2 (0.49) CACNA1HAOC3LTB4R2CNR2CNR1
SCHEMBL3824486 0.83 CACNA1H (0.41) CACNA1HAOC3LTB4R2CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed