SCHEMBL3824486

SCHEMBL3824486

CCN(CC)c1ccc(CN(C(=O)[C@@H](N)c2ccccc2)c2ccc(F)cc2)cn1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
AOC3 Q16853 1/20 0.40
MAPK14 Q16539 4/20 0.39
LTB4R2 Q9NPC1 3/20 0.39
CNR2 P34972 2/20 0.38
MMP1 P03956 2/20 0.38
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP13 P45452 2/20 0.38
CNR1 P21554 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
GRIA2 P42262 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825186 0.86 CACNA1H (0.44) CACNA1HAOC3MAPK14LTB4R2CNR2
SCHEMBL4736030 0.83 CACNA1H (0.47) CACNA1HAOC3MAPK14LTB4R2CNR2
SCHEMBL3823354 0.82 CACNA1H (0.40) CACNA1HTDP1AOC3MAPK14LTB4R2
SCHEMBL3820052 0.82 CACNA1H (0.40) CACNA1HTDP1AOC3MAPK14LTB4R2
SCHEMBL3071006 0.81 CACNA1H (0.47) CACNA1HAOC3MAPK14LTB4R2CNR2
SCHEMBL3815393 0.80 CACNA1H (0.45) CACNA1HAOC3LTB4R2CNR2CNR1
SCHEMBL3064331 0.78 CACNA1H (0.45) CACNA1HAOC3LTB4R2CNR2GRIA2
SCHEMBL3816063 0.77 CACNA1H (0.45) CACNA1HTDP1AOC3LTB4R2CNR2
SCHEMBL3063271 0.76 RIPK1 (0.49) CACNA1HAOC3LTB4R2CNR2GRIA2
Trifluoroacetic Acid SCHEMBL3054195 0.76 CACNA1H (0.42) CACNA1HAOC3LTB4R2CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091917-A1 ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-08-26 EP claimed
WO-2008073934-A1 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed