SCHEMBL4736233

SCHEMBL4736233

CN1CCCC[C@@H]1c1nc2cccnc2n1-c1ccc(C[C@H](NC(=O)c2c(Cl)cncc2Cl)C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 19/20 0.53
ITGB1 P05556 18/20 0.49
ITGB7 P26010 3/20 0.44
ITGB3 P05106 1/20 0.43
ITGAV P06756 1/20 0.43
ITGA5 P08648 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736084 0.86 ITGA4 (0.62) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4736103 0.86 ITGA4 (0.62) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4732547 0.86 ITGA4 (0.62) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4731194 0.82 ITGA4 (0.42) ITGA4ITGB1
SCHEMBL4734887 0.82 ITGA4 (0.42) ITGA4ITGB1
SCHEMBL4736591 0.80 ITGA4 (0.55) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4730816 0.80 ITGB1 (0.64) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4730854 0.80 ITGB1 (0.64) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4735439 0.80 ITGA4 (0.65) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4737750 0.79 ITGB1 (0.67) ITGA4ITGB1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed