SCHEMBL4736803

SCHEMBL4736803

O=C(/C=C/c1ccc(O)c(F)c1F)c1ccc(Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
CYP1B1 Q16678 1/20 0.50
DPP4 P27487 1/20 0.49
CXCL12 P48061 1/20 0.49
MAPT P10636 4/20 0.49
SNCA P37840 2/20 0.49
CHRNA7 P36544 1/20 0.49
CAPN1 P07384 1/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
RECQL P46063 2/20 0.47
RAB9A P51151 2/20 0.47
LMNA P02545 1/20 0.47
ALOX5 P09917 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736806 1.00 ESR1 (0.53) ESR1ESR2CYP1B1DPP4CXCL12
SCHEMBL4741756 0.79 GABRA3 (0.48) CYP1B1MAPTCHRNA7CAPN1CTSL
SCHEMBL4741758 0.79 GABRA3 (0.48) CYP1B1MAPTCHRNA7CAPN1CTSL
SCHEMBL4785911 0.79 DPP4 (0.55) ESR1ESR2CYP1B1DPP4CXCL12
SCHEMBL4785916 0.79 DPP4 (0.55) ESR1ESR2CYP1B1DPP4CXCL12
SCHEMBL29837090 0.76 MAPT (0.71) ESR1ESR2CYP1B1MAPTCHRNA7
SCHEMBL21647128 0.76 MAPT (0.71) ESR1ESR2CYP1B1MAPTCHRNA7
SCHEMBL21647129 0.76 MAPT (0.71) ESR1ESR2CYP1B1MAPTCHRNA7
SCHEMBL363885 0.76 CYP1B1 (0.51) ESR1ESR2CYP1B1DPP4MAPT
SCHEMBL16047829 0.75 MIF (0.56) ESR1ESR2DPP4MAPTSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087365-A2 SUBSTITUTED 1, 3-DIPHENYLPROPANE DERIVATIVES, PREPARATIONS AND USES OF SAME GENFIT (FR) 2008-07-24 WO disclosed
WO-2008087365-A2 SUBSTITUTED 1, 3-DIPHENYLPROPANE DERIVATIVES, PREPARATIONS AND USES OF SAME GENFIT (FR) 2008-07-24 WO disclosed