SCHEMBL4737097

SCHEMBL4737097

COc1ccc(CNc2nc(OCCCCC(=O)NO)nc3ccccc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.55
EGFR P00533 5/20 0.54
HDAC1 Q13547 5/20 0.54
HDAC8 Q9BY41 5/20 0.54
HDAC6 Q9UBN7 5/20 0.54
ERBB2 P04626 3/20 0.54
HDAC3 O15379 2/20 0.54
KDR P35968 2/20 0.54
HDAC4 P56524 2/20 0.54
HDAC7 Q8WUI4 2/20 0.54
HDAC2 Q92769 2/20 0.54
HDAC10 Q969S8 2/20 0.54
HDAC11 Q96DB2 2/20 0.54
HDAC9 Q9UKV0 2/20 0.54
HDAC5 Q9UQL6 2/20 0.54
POLB P06746 2/20 0.52
NR2F2 P24468 1/20 0.52
SLC2A1 P11166 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787621 0.99 EGFR (0.55) APPEGFRHDAC1HDAC8HDAC6
SCHEMBL4737141 0.99 EGFR (0.55) APPEGFRHDAC1HDAC8HDAC6
SCHEMBL4737772 0.84 SLC2A1 (0.57) APPHDAC1HDAC8HDAC6HDAC3
SCHEMBL4742773 0.84 SLC2A1 (0.57) APPHDAC1HDAC8HDAC6HDAC3
SCHEMBL4739328 0.84 SLC2A1 (0.57) APPHDAC1HDAC8HDAC6HDAC3
SCHEMBL3109840 0.82 APP (0.65) APPEGFRPOLBNR2F2SLC2A1
SCHEMBL3960300 0.81 LMNA (0.53) APPEGFRHDAC1HDAC8HDAC6
SCHEMBL3118629 0.80 APP (0.68) APPEGFRPOLBNR2F2SLC2A1
SCHEMBL3118894 0.80 APP (0.74) APPEGFRPOLBNR2F2SLC2A1
SCHEMBL3124803 0.80 APP (0.61) APPEGFRPOLBNR2F2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033747-A9 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS INC (MA) 2008-07-24 WO disclosed