SCHEMBL4737635

SCHEMBL4737635

O=C(Nc1oc(-c2ccccc2)nc1-c1ccccc1)c1ccccc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.54
KDR P35968 5/20 0.47
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
KCNK3 O14649 1/20 0.46
KCNK9 Q9NPC2 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
FLT1 P17948 1/20 0.45
FLT4 P35916 1/20 0.45
PTGS1 P23219 1/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MAPT P10636 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4260880 0.83 SMO (0.79) SMOKCNK3KCNK9MEN1KMT2A
SCHEMBL14148493 0.82 KDR (0.45) SMOKDRGAAFLT1FLT4
SCHEMBL4787849 0.81 ADCY1 (0.49) SMOKDRFLT1FLT4PTGS1
SCHEMBL14148814 0.81 SMO (0.67) SMOKDRFLT1FLT4SMN1; SMN2
SCHEMBL14148538 0.79 TP53 (0.57) SMOKDRMEN1KMT2AFLT1
SCHEMBL14148519 0.79 KDR (0.47) SMOKDRLMNAMEN1KMT2A
SCHEMBL4737638 0.79 KDR (0.55) KDRLMNAGAAMEN1KMT2A
SCHEMBL14148490 0.78 RXFP1 (0.53) SMOKDRLMNAGAARXFP1
SCHEMBL4741743 0.78 ADCY1 (0.65) LMNAGAAKCNK3PTGS1ALDH1A1
SCHEMBL14148837 0.78 KMT2A (0.60) KDRLMNAMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed