SCHEMBL4737704

SCHEMBL4737704

O=[N+]([O-])c1c(NCC2CC2)ccnc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.60
UTS2R Q9UKP6 2/20 0.44
PRKCQ Q04759 14/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2D6 P10635 2/20 0.38
DCLK1 O15075 1/20 0.38
MAP4K4 O95819 1/20 0.38
CDK1 P06493 1/20 0.38
PIM1 P11309 1/20 0.38
PRKACA P17612 1/20 0.38
CDK2 P24941 1/20 0.38
MATK P42679 1/20 0.38
FRK P42685 1/20 0.38
CSNK1D P48730 1/20 0.38
CLK2 P49760 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
IRAK1 P51617 1/20 0.38
RPS6KA3 P51812 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7034304 0.84 PTGER4 (0.43) PTGER4
SCHEMBL28076747 0.80 PTGER4 (0.41) PTGER4UTS2RKDM4C
SCHEMBL18285464 0.77 CUL4A (0.39) PTGER4CYP2C9
SCHEMBL28908277 0.76 KMT2A (0.53) CYP2C9CDK2GSK3AGSK3BCDK5
SCHEMBL13242139 0.76 KAT2B (0.40) PTGER4EGFRIGF1R
SCHEMBL19917187 0.75 KMT2A (0.56) CYP2C9CDK2GSK3AGSK3BCDK5
SCHEMBL15774396 0.75 PTGER4 (1.00) PTGER4PRKCQCYP3A4CYP2C9CYP2D6
SCHEMBL2572082 0.75 HTT (0.50) CYP3A4CYP2C9CYP2D6EGFRIGF1R
SCHEMBL12138409 0.74 ALDH1A1 (0.44)
SCHEMBL2708359 0.74 ALDH1A1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064830-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR PHARMACEUTICAL USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064830-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR PHARMACEUTICAL USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed