SCHEMBL473780

SCHEMBL473780

CN(C)C1CCCN(C(=O)c2ccc(-c3c(F)cnc4[nH]c5cnc(-c6cccnc6)cc5c34)cc2)C1.CN1CC(NC(=O)c2ccc(-c3c(F)cnc4[nH]c5cnc(-c6cccnc6)cc5c34)cc2)C1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATR Q13535 6/20 0.39
ALDH1A1 P00352 1/20 0.38
WNT1 P04628 3/20 0.38
DYRK1A Q13627 3/20 0.38
CHEK1 O14757 1/20 0.36
ACHE P22303 1/20 0.36
CDK1 P06493 3/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCND1 P24385 1/20 0.36
CCND3 P30281 1/20 0.36
CDK6 Q00534 1/20 0.36
JAK1 P23458 1/20 0.35
CDK2 P24941 2/20 0.35
PDE4B Q07343 1/20 0.35
MCHR1 Q99705 1/20 0.35
PIM1 P11309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11929486 0.93 ATR (0.43) ATRALDH1A1CHEK1ACHECDK1
SCHEMBL11929481 0.89 ATR (0.47) ATRCHEK1ACHECDK1CDK4
SCHEMBL11929488 0.89 ATR (0.47) ATRCHEK1ACHECDK1CDK4
SCHEMBL11908594 0.88 DYRK1A (0.43) WNT1DYRK1ACHEK1ACHEPIM1
SCHEMBL11909375 0.84 DYRK1A (0.53) ATRWNT1DYRK1ACHEK1ACHE
SCHEMBL473759 0.84 ATR (0.41) ATRCHEK1ACHECDK1CDK4
SCHEMBL3723614 0.83 CHEK1 (0.39) WNT1DYRK1ACHEK1ACHEPIM1
SCHEMBL11908845 0.81 RIPK1 (0.46) WNT1DYRK1ACHEK1ACHECDK2
SCHEMBL473748 0.81 CHEK1 (0.44) CHEK1ACHE
SCHEMBL11929463 0.81 RIPK1 (0.49) ATRCHEK1ACHECDK2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411389-A2 9H-PYRROLO[2,3-B: 5,4-C']DIPYRIDINE AZACARBOLINE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-02-01 EP claimed
WO-2010109084-A2 9H-PYRROLO[2,3-B: 5,4-C'] DIPYRIDINE AZACARBOLINE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-09-30 WO claimed