SCHEMBL4738162

SCHEMBL4738162

Nc1ncc(Cl)c(N2CCOC(CNC(=O)O)C2)c1[N+](=O)[O-]

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.35
CHEK2 O96017 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
GAA P10253 1/20 0.34
PPARA Q07869 1/20 0.34
MAPK1 P28482 1/20 0.34
KCNH2 Q12809 2/20 0.33
SMO Q99835 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2C9 P11712 1/20 0.33
ADRA2B P18089 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738167 1.00 CHEK1 (0.35) CHEK1CHEK2SMN1; SMN2GAAPPARA
SCHEMBL14163060 0.87 KCNH2 (0.36) CHEK1CHEK2SMN1; SMN2MAPK1KCNH2
SCHEMBL14162967 0.87 RPS6KB1 (0.35) CHEK1CHEK2SMN1; SMN2GAAKCNH2
SCHEMBL4738630 0.86 CHEK1 (0.38) CHEK1CHEK2SMN1; SMN2PPARAMAPK1
SCHEMBL4738164 0.80 ALDH1A1 (0.34) KMT2AMEN1LMNAMAPTRPS6KB1
SCHEMBL4735976 0.75 CHEK1 (0.38) CHEK1CHEK2PPARAMAPK1SMO
SCHEMBL2521642 0.71 GAA (0.39) GAAMAPK1CYP1A2CYP3A4CYP2C9
SCHEMBL14495694 0.69 HSP90AA1 (0.42) SMN1; SMN2GAAKMT2AMEN1LMNA
SCHEMBL15779396 0.68 KCNA5 (0.42) CHEK1CHEK2PPARAMAPK1MAPT
SCHEMBL209615 0.67 MAPT (0.45) SMN1; SMN2GAAKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075007-A1 MORPHOLINO-SUBSTITUTED BICYCLOHETEROARYL COMPOUNDS AND THEIR USE AS ANTI CANCER AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2008-06-26 WO disclosed