SCHEMBL4735976

SCHEMBL4735976

O=C(O)NCC1CN(c2c(Cl)cnc3[nH]c(=O)[nH]c23)CCO1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.38
CHEK2 O96017 3/20 0.38
AURKA O14965 3/20 0.36
AURKB Q96GD4 3/20 0.36
AKT1 P31749 1/20 0.35
PPARA Q07869 1/20 0.35
MAPK1 P28482 2/20 0.34
SLC34A1 Q06495 2/20 0.34
SMO Q99835 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14162815 0.87 CHEK1 (0.37) CHEK1CHEK2AURKAAURKBAKT1
SCHEMBL14162993 0.86 CHEK1 (0.37) CHEK1CHEK2AURKAAURKBAKT1
SCHEMBL4736887 0.85 CHEK1 (0.51) CHEK1CHEK2AKT1PPARAMAPK1
SCHEMBL4739231 0.85 CHEK1 (0.50) CHEK1CHEK2AKT1SLC34A1AKT2
SCHEMBL4736583 0.81 CHEK1 (0.46) CHEK1CHEK2AKT2
SCHEMBL4735981 0.80 AURKA (0.34) CHEK1CHEK2AURKAAURKB
SCHEMBL4737095 0.80 MAPK1 (0.39) CHEK1CHEK2AKT1PPARAMAPK1
SCHEMBL4738630 0.80 CHEK1 (0.38) CHEK1CHEK2PPARAMAPK1SMO
SCHEMBL4738167 0.75 CHEK1 (0.35) CHEK1CHEK2PPARAMAPK1SMO
SCHEMBL4738162 0.75 CHEK1 (0.35) CHEK1CHEK2PPARAMAPK1SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075007-A1 MORPHOLINO-SUBSTITUTED BICYCLOHETEROARYL COMPOUNDS AND THEIR USE AS ANTI CANCER AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2008-06-26 WO disclosed