SCHEMBL4738308

SCHEMBL4738308

CCOC(=O)C(Cc1c(C(=O)N(C)C)cc2c(nc(C)n2C)c1O)C(=O)c1c(C)cccc1C

nearest known ligand 0.31

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
CYP2D6 P10635 1/20 0.31
ACHE P22303 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
STAT6 P42226 1/20 0.30
KMT2A Q03164 1/20 0.30
HIF1A Q16665 1/20 0.30
ALOX5 P09917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739384 0.80 PARP1 (0.35) ALDH1A1
SCHEMBL4574787 0.73 MEN1 (0.33) ALDH1A1GAAKMT2A
SCHEMBL4963781 0.73 CTNNB1 (0.35) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL4965043 0.73 CTSA (0.33) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL4962044 0.73 CTSA (0.33) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL4962050 0.73 CTSA (0.33) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL4737338 0.71 KDM4E (0.36) KDM4EALDH1A1GAAKMT2A
SCHEMBL4738352 0.71 PARP1 (0.35) ALDH1A1
SCHEMBL5138943 0.70 CXCR2 (0.33) KDM4EALDH1A1HIF1A
SCHEMBL4664643 0.70 CXCR2 (0.33) KDM4EALDH1A1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074858-A1 INTERMEDIATES AND PROCESS FOR THE PRODUCTION OF 5-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES NYCOMED GMBH (DE) 2008-06-26 WO disclosed