SCHEMBL4738352

SCHEMBL4738352

Cc1ccccc1C(=O)C(Cc1c(C(=O)N(C)C)cc2c(nc(C3CC3)n2C)c1O)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
ALDH1A1 P00352 2/20 0.33
HSD17B10 Q99714 2/20 0.33
PKM P14618 1/20 0.33
ALOX15 P16050 1/20 0.32
AGTR1 P30556 1/20 0.32
AGTR2 P50052 1/20 0.32
TLR7 Q9NYK1 1/20 0.31
PDE9A O76083 3/20 0.31
CTSA P10619 1/20 0.31
PDE10A Q9Y233 1/20 0.31
BRD4 O60885 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739384 0.92 PARP1 (0.35) PARP1ALDH1A1HSD17B10PKMPDE9A
SCHEMBL4664629 0.79 ALDH1A1 (0.41) PARP1ALDH1A1HSD17B10PKMALOX15
SCHEMBL4664836 0.78 PARP1 (0.35) PARP1ALDH1A1HSD17B10PKMALOX15
SCHEMBL4963781 0.72 CTNNB1 (0.35) ALDH1A1HSD17B10BRD4
SCHEMBL4738308 0.71 CYP1A2 (0.31) ALDH1A1
SCHEMBL5666743 0.68 ALDH1A1 (0.34) PARP1ALDH1A1HSD17B10PKMALOX15
SCHEMBL4664618 0.67 KMT2A (0.35) ALDH1A1BRD4
Dimethylamine SCHEMBL5666747 0.67 PARP1 (0.35) PARP1ALDH1A1HSD17B10PKMALOX15
SCHEMBL4962044 0.66 CTSA (0.33) ALDH1A1HSD17B10CTSA
SCHEMBL4965043 0.66 CTSA (0.33) ALDH1A1HSD17B10CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074858-A1 INTERMEDIATES AND PROCESS FOR THE PRODUCTION OF 5-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES NYCOMED GMBH (DE) 2008-06-26 WO disclosed