SCHEMBL4739299

SCHEMBL4739299

CC1CC2(CCN1CC1CCC1)C(N[C@@H]1CC[Si](C)(C)C1)=NC(=O)N2c1cccc(F)c1

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.32
OPRM1 P35372 2/20 0.32
OPRL1 P41146 2/20 0.32
ADORA3 P0DMS8 2/20 0.31
ADORA1 P30542 2/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10262535 1.00 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL756766 1.00 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL755199 1.00 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL758140 1.00 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL757961 1.00 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
Hydrochloric Acid SCHEMBL755698 0.99 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
Hydrochloric Acid SCHEMBL759413 0.99 BACE1 (0.32) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL764691 0.88 ADORA3 (0.40) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL760030 0.84 BACE1 (0.34) BACE1OPRM1OPRL1ADORA3ADORA1
SCHEMBL755862 0.84 BACE1 (0.34) BACE1OPRM1OPRL1ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910364-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE Merck & Co., Inc. (US) 2008-04-16 EP claimed
WO-2007011833-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2007-01-25 WO claimed