SCHEMBL4739346

SCHEMBL4739346

O=c1[nH]c2c(O)ccc(CCNCCc3ccc([N+](=O)[O-])cc3)c2s1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 17/20 0.63
ADRB1 P08588 3/20 0.52
ABCB11 O95342 2/20 0.52
DRD2 P14416 1/20 0.52
PDE4A P27815 1/20 0.52
DRD3 P35462 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7839165 0.88 ABCB11 (0.64) ADRB2ADRB1ABCB11DRD2PDE4A
Hydrochloric Acid SCHEMBL7838052 0.87 ABCB11 (0.63) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL8528251 0.84 ABCB11 (0.73) ADRB2ADRB1ABCB11DRD2PDE4A
Hydrochloric Acid SCHEMBL8531813 0.84 ABCB11 (0.72) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL9522342 0.81 ADRB2 (0.72) ADRB2ADRB1ABCB11DRD2PDE4A
Hydrochloric Acid SCHEMBL8882013 0.80 ADRB2 (0.71) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL8879323 0.80 ADRB2 (0.61) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL9254881 0.80 ABCB11 (0.55) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL7841548 0.79 ADRB2 (0.61) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL9522645 0.79 ABCB11 (0.53) ADRB2ADRB1ABCB11DRD2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008096129-A1 NITROGEN CONTAINING HETROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA- 2 RECEPTORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed