SCHEMBL4739616

SCHEMBL4739616

Cc1nc(-c2ccc(C(F)(F)F)cc2)sc1C(=O)CCc1ccc(O)c(Cl)c1Cl

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
NPC1 O15118 1/20 0.55
GAA P10253 1/20 0.55
MAPT P10636 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HSP90AA1 P07900 1/20 0.48
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
PPARA Q07869 11/20 0.47
PPARD Q03181 5/20 0.47
PPARG P37231 5/20 0.47
FFAR1 O14842 2/20 0.44
NR1H4 Q96RI1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740491 0.88 ALDH1A1 (0.60) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4739681 0.88 MAPT (0.61) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4738839 0.88 NPC1 (0.57) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4740775 0.87 MAPT (0.44) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4738093 0.87 NPC1 (0.56) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4738817 0.86 ALDH1A1 (0.55) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4738885 0.85 MAPT (0.49) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4741834 0.84 ALDH1A1 (0.55) ALDH1A1NPC1GAAMAPTMEN1
SCHEMBL4741580 0.83 PPARA (0.56) ALDH1A1NPC1GAAPPARAPPARD
SCHEMBL4739607 0.82 PPARD (0.44) ALDH1A1NPC1GAAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087367-A2 SUBSTITUTED (PHENYLTHIAZOLYL)-PHENYL-PROPAN-1-ONE AND (PHENYLOXAZODYL)-PHENYL-PROPAN-1-ONE DERIVATIVES, PREPARATIONS AND USES OF SAME GENFIT (FR) 2008-07-24 WO disclosed
WO-2008087367-A2 SUBSTITUTED (PHENYLTHIAZOLYL)-PHENYL-PROPAN-1-ONE AND (PHENYLOXAZODYL)-PHENYL-PROPAN-1-ONE DERIVATIVES, PREPARATIONS AND USES OF SAME GENFIT (FR) 2008-07-24 WO disclosed