SCHEMBL4740819

SCHEMBL4740819

NC(=O)c1sc(-c2ccccc2)nc1-c1ccccc1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 7/20 0.85
DBF4 Q9UBU7 7/20 0.85
CCNE1 P24864 2/20 0.85
CDK2 P24941 2/20 0.85
PTGDR2 Q9Y5Y4 5/20 0.55
KDM4E B2RXH2 2/20 0.55
POLB P06746 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
ALDH1A1 P00352 3/20 0.53
MAPT P10636 2/20 0.53
GAA P10253 1/20 0.51
RARA P10276 1/20 0.51
RARB P10826 1/20 0.51
RARG P13631 1/20 0.51
HPGD P15428 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL974859 0.86 CDC7 (0.84) CDC7DBF4CCNE1CDK2PTGDR2
SCHEMBL9635836 0.83 CDC7 (0.61) CDC7DBF4CCNE1CDK2SMN1; SMN2
SCHEMBL3056066 0.83 CDC7 (0.65) CDC7DBF4CCNE1CDK2PTGDR2
SCHEMBL956697 0.83 CDC7 (0.61) CDC7DBF4CCNE1CDK2KDM4E
SCHEMBL2521905 0.83 ALDH1A1 (0.62) CDC7DBF4CCNE1CDK2KDM4E
SCHEMBL954078 0.82 CDC7 (0.68) CDC7DBF4CCNE1CDK2PTGDR2
SCHEMBL4243016 0.81 SMN1; SMN2 (0.76) CDC7DBF4CCNE1CDK2KDM4E
SCHEMBL15064348 0.80 CDC7 (0.62) CDC7DBF4CCNE1CDK2PTGDR2
SCHEMBL30511202 0.80 CDC7 (0.58) CDC7DBF4CCNE1CDK2PTGDR2
SCHEMBL975727 0.80 CDC7 (0.86) CDC7DBF4CCNE1CDK2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed