SCHEMBL4741114

SCHEMBL4741114

COC(=O)[C@](O)(c1ccccc1)C1CCCCC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.68
NFE2L2 Q16236 1/20 0.68
POLB P06746 1/20 0.64
ALDH1A1 P00352 2/20 0.63
CHRM3 P20309 5/20 0.61
CHRM2 P08172 4/20 0.61
CHRM1 P11229 3/20 0.61
KCNH2 Q12809 3/20 0.61
SLC6A3 Q01959 2/20 0.61
CHRM4 P08173 2/20 0.60
CHRM5 P08912 2/20 0.60
HTR2B P41595 2/20 0.60
CYP1A2 P05177 2/20 0.60
HRH1 P35367 1/20 0.60
CYP3A4 P08684 2/20 0.59
CYP2D6 P10635 2/20 0.59
CYP2C19 P33261 2/20 0.58
CYP2C9 P11712 1/20 0.58
PKM P14618 1/20 0.58
NFKB1 P19838 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27483674 1.00 KEAP1 (0.68) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL1610849 1.00 KEAP1 (0.68) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL1234889 0.98 KEAP1 (0.70) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL522945 0.98 KEAP1 (0.70) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL2062807 0.98 KEAP1 (0.70) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL10842570 0.93 KEAP1 (0.62) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL403319 0.86 KEAP1 (0.66) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL13574070 0.85 CHRM2 (0.70) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL13574067 0.85 CHRM2 (0.70) KEAP1NFE2L2POLBALDH1A1CHRM3
SCHEMBL290176 0.85 CHRM2 (0.70) KEAP1NFE2L2POLBALDH1A1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008096127-A2 BICYCLO[2.2.1]HEPT-7-YLAMINE DERIVATIVES AND THEIR USE AS M3 MUSCARINIC RECEPTOR MODULATORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed