SCHEMBL4741154

SCHEMBL4741154

CN(CCc1cnc(C(O)(c2ccccc2)C2CCCCC2)o1)Cc1cccc(CCO)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 10/20 0.35
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RECQL P46063 1/20 0.33
POLB P06746 1/20 0.32
CHRM2 P08172 9/20 0.32
CHRM4 P08173 9/20 0.32
CHRM5 P08912 9/20 0.32
CHRM1 P11229 9/20 0.32
KDM4E B2RXH2 2/20 0.32
CYP2J2 P51589 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741153 1.00 CHRM3 (0.35) CHRM3NR1H2NR1H3ALDH1A1CYP2D6
SCHEMBL3224220 0.92 CHRM3 (0.36) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3232872 0.92 CHRM3 (0.36) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3226330 0.91 CHRM3 (0.39) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3226320 0.91 CHRM3 (0.39) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3236054 0.87 ACHE (0.37) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3236047 0.87 ACHE (0.37) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3234490 0.83 CHRM3 (0.35) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL3234494 0.83 CHRM3 (0.35) CHRM3ALDH1A1POLBCHRM2CHRM4
SCHEMBL1109856 0.82 POLB (0.44) CHRM3ALDH1A1CYP2D6POLBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008096129-A1 NITROGEN CONTAINING HETROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA- 2 RECEPTORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed