SCHEMBL4741246

SCHEMBL4741246

Nc1nc2c(c(-c3ccccc3)n1)-c1cc(N)c(Cl)cc1CC2

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.42
ADORA1 P30542 15/20 0.42
ADORA2A P29274 15/20 0.42
ADORA2B P29275 2/20 0.41
P2RX7 Q99572 1/20 0.38
PDE4B Q07343 1/20 0.37
NUDT1 P36639 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741259 0.89 TYMS (0.41) TYMSADORA1ADORA2AADORA2BKDM4E
SCHEMBL4740440 0.88 TYMS (0.41) TYMSADORA1ADORA2AADORA2BKDM4E
SCHEMBL4737740 0.87 ADORA2A (0.46) TYMSADORA1ADORA2AADORA2BKDM4E
SCHEMBL4741251 0.87 ADORA2A (0.43) TYMSADORA1ADORA2AADORA2BKDM4E
SCHEMBL4739911 0.85 TYMS (0.52) TYMSADORA1ADORA2AADORA2B
SCHEMBL4741224 0.84 HRH3 (0.53) TYMSADORA1ADORA2AKDM4EALDH1A1
SCHEMBL4740434 0.84 ADORA2A (0.51) TYMSADORA1ADORA2AADORA2BKDM4E
SCHEMBL4740744 0.83 TYMS (0.40) TYMSADORA1ADORA2APDE4BKDM4E
SCHEMBL4738543 0.83 MAP2K4 (0.41) TYMSP2RX7PDE4B
SCHEMBL14148131 0.83 TYMS (0.38) TYMSADORA1ADORA2AADORA2BP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed