SCHEMBL4740440

SCHEMBL4740440

Nc1nc2c(c(-c3ccc(F)cc3)n1)-c1cc(N)c(Cl)cc1CC2

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.41
ADORA2A P29274 14/20 0.37
ADORA1 P30542 13/20 0.37
ADORA2B P29275 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
HRH2 P25021 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
PIKFYVE Q9Y2I7 1/20 0.36
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741246 0.88 TYMS (0.42) TYMSADORA2AADORA1ADORA2BKDM4E
SCHEMBL4741251 0.87 ADORA2A (0.43) TYMSADORA2AADORA1ADORA2BKDM4E
SCHEMBL4741259 0.86 TYMS (0.41) TYMSADORA2AADORA1ADORA2BHRH2
SCHEMBL4737447 0.86 TYMS (0.38) TYMSADORA2AADORA1
SCHEMBL4736837 0.86 TYMS (0.38) TYMSADORA2AADORA1ADORA2BADORA3
SCHEMBL4787500 0.85 TYMS (0.50) TYMSADORA2AADORA1ADORA2BADORA3
SCHEMBL4741224 0.85 HRH3 (0.53) TYMSADORA2AADORA1HRH2HRH3
SCHEMBL4740744 0.84 TYMS (0.40) TYMSADORA2AADORA1KDM4E
SCHEMBL4741116 0.83 DHFR (0.40) TYMSADORA2AADORA1
SCHEMBL4737740 0.80 ADORA2A (0.46) TYMSADORA2AADORA1ADORA2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed