SCHEMBL4737740

SCHEMBL4737740

Nc1nc2c(c(-c3cccnc3)n1)-c1cc(N)c(Cl)cc1CC2

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.46
NQO2 P16083 3/20 0.46
ADORA2B P29275 3/20 0.46
ADORA1 P30542 4/20 0.40
HRH3 Q9Y5N1 1/20 0.40
TYMS P04818 1/20 0.39
CYP11B1 P15538 5/20 0.38
CYP11B2 P19099 5/20 0.38
CYP1A2 P05177 2/20 0.38
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
PTK2 Q05397 1/20 0.36
CYP2A6 P11509 1/20 0.36
BRAF P15056 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741246 0.87 TYMS (0.42) ADORA2AADORA2BADORA1TYMSKDM4E
SCHEMBL4741259 0.86 TYMS (0.41) ADORA2ANQO2ADORA2BADORA1HRH3
SCHEMBL4741251 0.82 ADORA2A (0.43) ADORA2AADORA2BADORA1TYMSKDM4E
SCHEMBL14147950 0.81 MEN1 (0.40) ADORA2ANQO2ADORA2BADORA1CYP11B1
SCHEMBL4740440 0.80 TYMS (0.41) ADORA2AADORA2BADORA1HRH3TYMS
SCHEMBL4740434 0.79 ADORA2A (0.51) ADORA2AADORA2BADORA1HRH3TYMS
SCHEMBL4738543 0.78 MAP2K4 (0.41) TYMS
SCHEMBL4736829 0.78 JAK2 (0.39) ADORA2AADORA1TYMS
SCHEMBL4741224 0.77 HRH3 (0.53) ADORA2AADORA1HRH3TYMSKDM4E
SCHEMBL4786839 0.77 PIKFYVE (0.39) ADORA2ATYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed