SCHEMBL4743802

SCHEMBL4743802

COc1ccc(CN2CCN(CCCCCOc3ccc(C(=O)c4ccc(Cl)cc4)cc3)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.66
KCNA5 P22460 1/20 0.61
DRD3 P35462 1/20 0.61
HRH1 P35367 2/20 0.59
HRH2 P25021 1/20 0.59
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
LMNA P02545 1/20 0.57
HRH3 Q9Y5N1 10/20 0.57
HRH4 Q9H3N8 1/20 0.57
POLB P06746 1/20 0.55
RECQL P46063 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
BCHE P06276 1/20 0.54
ACHE P22303 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743805 0.89 KDM4E (0.69) HRH1KDM4EALDH1A1MEN1KMT2A
SCHEMBL4746670 0.84 HRH3 (0.54) DRD2HRH1KDM4EALDH1A1MEN1
SCHEMBL7367224 0.83 HRH3 (0.81) KDM4EALDH1A1MEN1KMT2AHRH3
SCHEMBL28813326 0.82 DRD3 (0.65) DRD2KCNA5DRD3ALDH1A1MEN1
SCHEMBL4743801 0.82 HRH3 (0.59) DRD2HRH1MEN1KMT2AHRH3
SCHEMBL4743140 0.82 HRH3 (0.65) DRD2KCNA5HRH1KDM4EALDH1A1
SCHEMBL4746238 0.82 HRH3 (0.65) HRH1KDM4EALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL7371901 0.82 HRH3 (0.79) KDM4EALDH1A1MEN1KMT2AHRH3
SCHEMBL4746235 0.81 HRH3 (0.55) DRD2HRH1MEN1KMT2AHRH3
SCHEMBL4746696 0.80 HRH3 (0.57) DRD2HRH1MEN1KMT2AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107320-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed