SCHEMBL4743844

SCHEMBL4743844

CCOC(=O)c1sc(C)nc1-c1cccc(C)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
HSD17B10 Q99714 2/20 0.57
HPGD P15428 2/20 0.55
DHODH Q02127 8/20 0.53
CDC7 O00311 4/20 0.53
DBF4 Q9UBU7 4/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
TRPM8 Q7Z2W7 3/20 0.49
GSTO1 P78417 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
MAPT P10636 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1340195 0.87 TRPM8 (0.65) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL1966336 0.87 DHODH (0.59) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL1968418 0.87 TRPM8 (0.65) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL11164259 0.87 ALDH1A1 (0.77) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL11281010 0.87 ALDH1A1 (0.55) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL8823153 0.86 ALDH1A1 (0.75) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL1970502 0.84 MAPT (0.67) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL1968834 0.83 TRPM8 (0.60) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL6766164 0.83 DHODH (0.60) ALDH1A1HSD17B10HPGDDHODHCDC7
SCHEMBL1398685 0.82 MAPK14 (0.52) ALDH1A1DHODHCDC7DBF4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087611-A2 PYRROLIDINE- AND PIPERIDINE- BIS-AMIDE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-24 WO disclosed