SCHEMBL4744462

SCHEMBL4744462

O=C(CN1CCN(CCCCCOc2ccc3c(-c4ccc(Cl)cc4)coc3c2)CC1)NCC1CCCCC1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.51
AVPR1B P47901 2/20 0.49
SIGMAR1 Q99720 1/20 0.48
BCHE P06276 2/20 0.44
ACHE P22303 2/20 0.44
MAOB P27338 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744422 0.96 AVPR1B (0.52) HRH3AVPR1BSIGMAR1
SCHEMBL4741958 0.89 HRH3 (0.53) HRH3SIGMAR1BCHEACHE
SCHEMBL4744392 0.88 HRH3 (0.58) HRH3BCHEACHEMAOB
SCHEMBL4742594 0.88 HRH3 (0.56) HRH3BCHEACHEMAOB
SCHEMBL4742644 0.87 HRH3 (0.52) HRH3SIGMAR1BCHEACHE
SCHEMBL4743420 0.87 HRH3 (0.51) HRH3AVPR1BSIGMAR1BCHEACHE
SCHEMBL4742556 0.86 HRH3 (0.54) HRH3SIGMAR1BCHEACHE
SCHEMBL4741928 0.86 HRH3 (0.54) HRH3SIGMAR1BCHEACHE
SCHEMBL4744494 0.85 HRH3 (0.50) HRH3SIGMAR1BCHEACHE
SCHEMBL4744473 0.85 HRH3 (0.50) HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107321-A1 HETEROCYCLIC COMPOUNDS USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO claimed
WO-2008107321-A1 HETEROCYCLIC COMPOUNDS USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed