SCHEMBL4744522

SCHEMBL4744522

O=C(O)C1CCCCN1Cc1cccc(OCc2coc(-c3ccc(C(F)(F)F)cc3)n2)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.56
PPARG P37231 3/20 0.56
CD274 Q9NZQ7 5/20 0.53
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALOX5AP P20292 4/20 0.44
SPHK1 Q9NYA1 1/20 0.43
PDCD1 Q15116 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743974 0.98 PPARA (0.57) PPARAPPARGCD274POLBALDH1A1
SCHEMBL4743964 0.98 PPARA (0.57) PPARAPPARGCD274POLBALDH1A1
SCHEMBL4748089 0.92 PPARA (0.58) PPARAPPARGCD274POLBALDH1A1
SCHEMBL4745017 0.91 CD274 (0.62) PPARACD274POLBSPHK1PDCD1
SCHEMBL4747149 0.90 KDM4E (0.49) PPARAPPARGCD274ALDH1A1ALOX5AP
SCHEMBL4787471 0.90 CD274 (0.59) PPARAPPARGCD274POLBSPHK1
SCHEMBL4747119 0.89 PPARA (0.59) PPARAPPARGCD274POLBALDH1A1
SCHEMBL4744260 0.89 CD274 (0.59) PPARAPPARGCD274POLBSPHK1
SCHEMBL4744265 0.89 CD274 (0.59) PPARAPPARGCD274POLBSPHK1
SCHEMBL4747069 0.88 HRH3 (0.47) PPARAPPARGCD274ALDH1A1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO claimed
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO disclosed