SCHEMBL4744531

SCHEMBL4744531

CC(O)COc1ccc(C(NC(=O)OC(C)(C)C)C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.50
CTSK P43235 1/20 0.50
GPR88 Q9GZN0 8/20 0.48
LMNA P02545 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
S1PR3 Q99500 1/20 0.42
ATM Q13315 1/20 0.42
MAPT P10636 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
PPARA Q07869 2/20 0.40
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379296 1.00 CTSS (0.50) CTSSCTSKGPR88LMNAITGB3
SCHEMBL3379292 1.00 CTSS (0.50) CTSSCTSKGPR88LMNAITGB3
SCHEMBL3379286 1.00 CTSS (0.50) CTSSCTSKGPR88LMNAITGB3
SCHEMBL1554766 0.88 GPR88 (0.54) CTSSCTSKGPR88
SCHEMBL1554764 0.88 GPR88 (0.54) CTSSCTSKGPR88
SCHEMBL1554765 0.88 GPR88 (0.54) CTSSCTSKGPR88
SCHEMBL2500015 0.88 GPR88 (0.54) CTSSCTSKGPR88
SCHEMBL1584437 0.86 GPR88 (0.65) GPR88
SCHEMBL3377050 0.86 CTSS (0.53) CTSSCTSKGPR88LMNAITGB3
SCHEMBL3377047 0.86 CTSS (0.53) CTSSCTSKGPR88LMNAITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1989186-A1 HYDANTOIN BASED KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2008-11-12 EP disclosed
WO-2008101840-A1 COMBINATION OF ERLOTINIB AND MEK-INHIBITORS FOR INHIBITING PROLIFERATION OF TUMOR CELLS F. HOFFMANN-LA ROCHE AG (CH) 2008-08-28 WO disclosed
WO-2007096259-A1 HYDANTOIN BASED KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-30 WO disclosed