SCHEMBL4744629

SCHEMBL4744629

Cc1oc(-c2ccccc2)nc1COc1cccc(COC(=O)C2CCCN2)c1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.62
PPARG P37231 17/20 0.53
PPARA Q07869 17/20 0.53
FFAR1 O14842 1/20 0.51
CYP2C9 P11712 1/20 0.49
KCNH2 Q12809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743666 0.98 KDR (0.60) KDRPPARGPPARAFFAR1CYP2C9
SCHEMBL4743931 0.97 KDR (0.61) KDRPPARGPPARAFFAR1CYP2C9
SCHEMBL4748548 0.94 PPARG (0.55) KDRPPARGPPARACYP2C9KCNH2
SCHEMBL4744642 0.90 PPARG (0.55) KDRPPARGPPARACYP2C9KCNH2
SCHEMBL4743967 0.86 PPARA (0.49) KDRPPARGPPARACYP2C9KCNH2
SCHEMBL4744698 0.86 FFAR1 (0.63) KDRPPARGPPARAFFAR1
SCHEMBL4748098 0.86 PPARA (0.52) PPARGPPARA
SCHEMBL4747104 0.84 PPARA (0.48) KDRPPARGPPARACYP2C9KCNH2
SCHEMBL27650834 0.83 KDR (0.74) KDRPPARGPPARAFFAR1CYP2C9
SCHEMBL4745030 0.82 PPARG (0.59) PPARGPPARAFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO disclosed