SCHEMBL4745320

SCHEMBL4745320

Cc1cc(O)c2cc(N3CCN(C)CC3)ccc2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
ADRA2A P08913 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
IDO1 P14902 2/20 0.51
TDO2 P48775 2/20 0.51
IDO2 Q6ZQW0 2/20 0.51
MEN1 O00255 1/20 0.50
GLA P06280 1/20 0.50
GAA P10253 1/20 0.50
KMT2A Q03164 1/20 0.50
DNMT1 P26358 1/20 0.50
RAD52 P43351 1/20 0.50
ALDH1A1 P00352 2/20 0.45
HTR6 P50406 2/20 0.45
TOP1 P11387 2/20 0.45
TOP2A P11388 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30594984 0.84 ADRB1 (0.53) KDM4EIDO1TDO2IDO2HTR6
SCHEMBL29125442 0.84 KMT2A (0.57) KDM4ESMN1; SMN2NPC1RAB9ATDO2
SCHEMBL4745451 0.83 KDM4E (0.56) KDM4ESMN1; SMN2NPC1RAB9AADRA2A
SCHEMBL27909494 0.81 KDM4E (0.48) KDM4ESMN1; SMN2NPC1RAB9AIDO1
SCHEMBL29125356 0.78 MAPT (0.49) SMN1; SMN2MEN1KMT2AALDH1A1MAPT
SCHEMBL30594931 0.78 MAPT (0.49) SMN1; SMN2MEN1KMT2AALDH1A1MAPT
SCHEMBL13312472 0.76 AURKA (0.53) KDM4ESMN1; SMN2NPC1RAB9AIDO1
SCHEMBL25746316 0.74 KDM4E (0.56) KDM4ESMN1; SMN2NPC1RAB9AADRA2A
SCHEMBL27170983 0.74 KDM4E (0.56) KDM4ESMN1; SMN2NPC1RAB9AADRA2A
SCHEMBL11762820 0.74 KDM4E (0.45) KDM4ESMN1; SMN2NPC1RAB9AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117079-A1 ANTIMICROBIAL COMPOUNDS BASED UPON 4-AMINOQUINOLINE HELPERBY THERAPEUTICS LIMITED (GB) 2008-10-02 WO disclosed