SCHEMBL4745458

SCHEMBL4745458

NC(=O)Nc1ncnc2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.65
LMNA P02545 2/20 0.58
ALDH1A1 P00352 1/20 0.54
EGFR P00533 4/20 0.53
ABCG2 Q9UNQ0 3/20 0.53
DAPK3 O43293 1/20 0.53
MAP4K4 O95819 1/20 0.53
ABL1 P00519 1/20 0.53
ERBB2 P04626 1/20 0.53
PIM1 P11309 1/20 0.53
PRKACA P17612 1/20 0.53
LTK P29376 1/20 0.53
MAPK8 P45983 1/20 0.53
CSNK1A1 P48729 1/20 0.53
RPS6KA3 P51812 1/20 0.53
LIMK1 P53667 1/20 0.53
MAP2K1 Q02750 1/20 0.53
ACVR1 Q04771 1/20 0.53
TYRO3 Q06418 1/20 0.53
MAP4K2 Q12851 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31004010 1.00 ADORA3 (0.65) ADORA3LMNAALDH1A1EGFRABCG2
SCHEMBL4751092 0.83 ADORA3 (0.56) ADORA3LMNAALDH1A1EGFRABCG2
SCHEMBL28645156 0.83 ADORA3 (0.65) ADORA3LMNAALDH1A1EGFRABCG2
SCHEMBL4424939 0.83 ADORA3 (0.56) ADORA3LMNAALDH1A1EGFRABCG2
SCHEMBL31060719 0.79 ADORA3 (1.00) ADORA3LMNAEGFRABCG2DAPK3
SCHEMBL4689838 0.79 ADORA3 (1.00) ADORA3LMNAEGFRABCG2DAPK3
SCHEMBL18552030 0.76 EGFR (0.61) ADORA3LMNAALDH1A1EGFRABCG2
SCHEMBL30317647 0.76 EGFR (0.61) ADORA3LMNAEGFRABCG2DAPK3
SCHEMBL3874722 0.76 EGFR (0.61) ADORA3LMNAEGFRABCG2DAPK3
SCHEMBL21879270 0.75 ALDH1A1 (0.57) ADORA3LMNAALDH1A1EGFRABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296973-B1 GUANIDINE DERIVATIVES OF QUINAZOLINE FOR USE IN THE TREATMENT OF AUTOIMMUNE DISEASES ASTRAZENECA AB (SE) 2008-11-05 EP disclosed