SCHEMBL4745571

SCHEMBL4745571

Cc1nn(-c2ccccn2)c(O)c1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC11A2 P49281 3/20 0.54
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44
MAPT P10636 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
ALOX15 P16050 1/20 0.42
HTT P42858 2/20 0.42
XBP1 P17861 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
AVPR1A P37288 2/20 0.41
OXTR P30559 1/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
BACE1 P56817 1/20 0.41
CCNA2 P20248 3/20 0.41
CDK2 P24941 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690425 0.87 SLC11A2 (0.55) SLC11A2PDCD1CD274MAPTALDH1A1
SCHEMBL3682387 0.86 SLC11A2 (0.51) SLC11A2MAPTALDH1A1HPGDHSD17B10
SCHEMBL4746341 0.85 ALDH1A1 (0.48) SLC11A2MAPTALDH1A1HPGDHSD17B10
SCHEMBL3692788 0.83 MAPT (0.48) SLC11A2MAPTALDH1A1HPGDHSD17B10
SCHEMBL3689323 0.81 FFAR4 (0.45) MAPTALDH1A1HPGDHSD17B10ALOX15
SCHEMBL3683176 0.81 SLC11A2 (0.53) SLC11A2PDCD1CD274MAPTALDH1A1
SCHEMBL3683062 0.80 MAPT (0.52) SLC11A2MAPTALDH1A1HPGDHSD17B10
SCHEMBL3681849 0.80 SLC11A2 (0.54) SLC11A2MAPTALDH1A1HPGDHSD17B10
SCHEMBL3683412 0.79 MAPT (0.45) SLC11A2MAPTALDH1A1HPGDHSD17B10
SCHEMBL3693842 0.78 MEN1 (0.42) MAPTALDH1A1HPGDHSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008121861-A2 PYRAZOLE AND PYRROLE COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-10-09 WO claimed
WO-2008121861-A2 PYRAZOLE AND PYRROLE COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-10-09 WO disclosed
WO-2008121861-A2 PYRAZOLE AND PYRROLE COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-10-09 WO disclosed