SCHEMBL4745908

SCHEMBL4745908

O=C1CSC(c2cccc(Br)c2)N1c1ccc(Oc2ccc(Cl)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.63
CA2 P00918 4/20 0.63
CA9 Q16790 4/20 0.63
KMT2A Q03164 1/20 0.55
ALDH1A1 P00352 1/20 0.54
HTT P42858 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
GFER P55789 3/20 0.53
MAPT P10636 1/20 0.49
METAP1 P53582 1/20 0.47
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47
TUBB2A Q13885 1/20 0.47
TUBB8 Q3ZCM7 1/20 0.47
TUBA3E Q6PEY2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743966 0.90 CA1 (0.53) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4748024 0.90 CA1 (0.67) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4747965 0.88 KMT2A (0.56) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4743949 0.88 ALDH1A1 (0.64) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4743914 0.87 ALDH1A1 (0.50) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4745883 0.87 KMT2A (0.55) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4747343 0.87 KMT2A (0.58) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4743906 0.87 CA1 (0.57) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4743907 0.87 KMT2A (0.55) CA1CA2CA9KMT2AALDH1A1
SCHEMBL4743528 0.87 KMT2A (0.74) CA1CA2CA9KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO claimed
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO disclosed