SCHEMBL474607

SCHEMBL474607

CC(=O)C1(C(=O)O)CCCN1c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.44
CYP2C19 P33261 6/20 0.44
HIF1A Q16665 2/20 0.44
USP2 O75604 4/20 0.43
ALDH1A1 P00352 3/20 0.42
MAPK1 P28482 3/20 0.42
FFAR1 O14842 1/20 0.40
BDKRB2 P30411 1/20 0.40
CYP1A2 P05177 4/20 0.39
CYP2C9 P11712 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HSD17B10 Q99714 3/20 0.39
TSHR P16473 2/20 0.39
CYP2D6 P10635 2/20 0.39
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360954 0.85 DRD2 (0.40) CYP3A4CYP2C19HIF1AUSP2ALDH1A1
SCHEMBL27627652 0.83 CYP2C19 (0.38) CYP3A4CYP2C19HIF1AUSP2ALDH1A1
SCHEMBL27508208 0.80 FFAR1 (0.38) CYP3A4CYP2C19HIF1AUSP2ALDH1A1
SCHEMBL16760058 0.78 AKR1C3 (0.43) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL15059997 0.78 FFAR1 (0.44) CYP3A4CYP2C19HIF1AUSP2ALDH1A1
SCHEMBL11250730 0.76 METAP2 (0.41) FFAR1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL2899064 0.76 CYP3A4 (0.40) CYP3A4CYP2C19HIF1AUSP2ALDH1A1
SCHEMBL3836402 0.75 CYP3A4 (0.39) CYP3A4CYP2C19HIF1AUSP2ALDH1A1
SCHEMBL2733709 0.73 NR1H2 (0.52) CYP3A4CYP2C19HIF1AALDH1A1FFAR1
SCHEMBL2733711 0.73 NR1H2 (0.52) CYP3A4CYP2C19HIF1AALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651342-A The inhibitor of hepatitis c viral replication 默沙东公司 2019-04-19 CN disclosed
CN-103880862-B The inhibitor of hepatitis c viral replication 默沙东公司 2018-09-25 CN disclosed
CN-102427729-A Inhibitors of hepatitis c virus replication MERCK SHARP & DOHME 2012-04-25 CN disclosed
EP-2410844-A1 INHIBITORS OF HEPATITIS C VIRUS REPLICATION Merck Sharp & Dohme Corp. (US) 2012-02-01 EP disclosed
WO-2010111483-A1 INHIBITORS OF HEPATITIS C VIRUS REPLICATION MERCK SHARP & DOHME CORP. (US) 2010-09-30 WO disclosed