SCHEMBL4746682

SCHEMBL4746682

FC#Cc1ccc(F)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GRM5 P41594 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
NR3C2 P08235 1/20 0.38
IDO1 P14902 2/20 0.38
AGXT P21549 2/20 0.38
MME P08473 1/20 0.37
ECE1 P42892 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
CA3 P07451 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
TRPV4 Q9HBA0 1/20 0.34
NFE2L2 Q16236 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3245685 0.87 ALDH1A1 (0.46) ALDH1A1ATMTDP1GRM5PTGDR2
SCHEMBL6141336 0.79 ALDH1A1 (0.39) ALDH1A1ATMTDP1GRM5PTGDR2
SCHEMBL4231062 0.79 NR3C2 (0.40) ALDH1A1ATMTDP1GRM5PTGDR2
SCHEMBL6364007 0.74 TRPV3 (0.39) ALDH1A1GRM5PTGDR2NR3C2MME
SCHEMBL29896412 0.74 TRPV3 (0.39) ALDH1A1GRM5PTGDR2NR3C2MME
SCHEMBL29305005 0.74 TRPV3 (0.41) ALDH1A1ATMTDP1GRM5PTGDR2
SCHEMBL79584 0.74 MME (0.46) ALDH1A1GRM5PTGDR2NR3C2MME
SCHEMBL14770099 0.74 ALDH1A1 (0.35) ALDH1A1ATMTDP1GRM5PTGDR2
SCHEMBL2764279 0.73 ALDH1A1 (0.42) ALDH1A1ATMTDP1GRM5PTGDR2
SCHEMBL22616325 0.73 ALDH1A1 (0.42) ALDH1A1ATMTDP1GRM5PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651621-B1 2- (QUINOXALIN-5-YLSULFONYLAMINO) -BENZAMIDE COMPOUNDS AS CCK2 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2008-08-06 EP claimed