SCHEMBL4747788

SCHEMBL4747788

N#Cc1c[nH]c2ncc(-c3cccc(NC(=O)CN4CCOCC4)c3)cc12

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.56
MAP4K4 O95819 1/20 0.56
PLCG1 P19174 2/20 0.54
BTK Q06187 7/20 0.52
ITK Q08881 7/20 0.52
ALDH1A1 P00352 5/20 0.49
HTT P42858 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
MAPK1 P28482 1/20 0.47
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746451 0.78 BTK (0.56) PLCG1BTKITK
SCHEMBL16176821 0.75 BTK (0.76) JAK3PLCG1BTKITK
SCHEMBL14069150 0.73 BTK (0.50) PLCG1BTKITK
SCHEMBL1463453 0.72 JAK3 (1.00) JAK3MAP4K4ALDH1A1HTTMEN1
SCHEMBL15587657 0.72 MAP4K4 (1.00) MAP4K4
SCHEMBL4746500 0.71 TNIK (0.58) SMN1; SMN2
SCHEMBL12746101 0.71 SMN1; SMN2 (0.64) JAK3MAP4K4ALDH1A1HTTMEN1
SCHEMBL17938939 0.70 PLCG1 (1.00) PLCG1BTKITK
SCHEMBL17938942 0.70 PLCG1 (1.00) PLCG1BTKITK
SCHEMBL16176566 0.70 BTK (0.77) PLCG1BTKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO claimed
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO disclosed
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO disclosed