SCHEMBL4746451

SCHEMBL4746451

N#Cc1c[nH]c2ncc(-c3cccc(NC(=O)CCNC(=O)O)c3)cc12

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 12/20 0.56
ITK Q08881 11/20 0.56
PLCG1 P19174 2/20 0.49
RIPK1 Q13546 2/20 0.48
IGF1R P08069 2/20 0.48
NTRK1 P04629 1/20 0.46
CDK8 P49336 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743377 0.89 PRMT5 (0.46) BTKITKRIPK1IGF1RCDK8
SCHEMBL14069150 0.87 BTK (0.50) BTKITKPLCG1NTRK1CDK8
SCHEMBL4747788 0.78 JAK3 (0.56) BTKITKPLCG1
SCHEMBL14069152 0.76 PRMT5 (0.42) BTKITKCDK8
SCHEMBL16176821 0.75 BTK (0.76) BTKITKPLCG1RIPK1IGF1R
SCHEMBL4746500 0.74 TNIK (0.58) NTRK1
SCHEMBL21118214 0.72 BTK (0.82) BTKITKPLCG1RIPK1IGF1R
SCHEMBL16176744 0.72 BTK (1.00) BTKITKPLCG1RIPK1IGF1R
SCHEMBL4747692 0.71 TNIK (0.63) ITKRIPK1NTRK1
SCHEMBL4166436 0.71 AXL (0.55) BTKITKPLCG1RIPK1IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO claimed
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO disclosed