SCHEMBL4748773

SCHEMBL4748773

O=C(C=Cc1ccc(O)cc1)c1cccc(Nc2ccnc3cc(Cl)ccc23)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.59
MAPT P10636 1/20 0.59
ATM Q13315 1/20 0.59
CYP2D6 P10635 6/20 0.52
CYP1A2 P05177 5/20 0.52
APP P05067 2/20 0.47
NR4A2 P43354 2/20 0.47
FADS1 O60427 1/20 0.47
KCNH2 Q12809 3/20 0.46
PTGS2 P35354 2/20 0.46
ABCB11 O95342 1/20 0.46
CHRM2 P08172 1/20 0.46
HTR1A P08908 1/20 0.46
CHRM1 P11229 1/20 0.46
DRD2 P14416 1/20 0.46
ADRA2C P18825 1/20 0.46
SLC6A2 P23975 1/20 0.46
OPRM1 P35372 1/20 0.46
HTR2B P41595 1/20 0.46
CYP2J2 P51589 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14024396 0.95 CYP2D6 (0.52) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4748788 0.95 CYP2D6 (0.52) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL30383538 0.90 GAA (0.59) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024410 0.90 GAA (0.59) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024471 0.87 APP (0.46) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4748784 0.85 CYP2D6 (0.52) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4748929 0.84 MAPT (0.60) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024382 0.84 MAPT (0.60) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4748932 0.84 MAPT (0.60) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024514 0.81 CXCL12 (0.52) GAACYP2D6CYP1A2APPNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed